( 50 of 255506 ) |
United States Patent | 7,968,752 |
Lee , et al. | June 28, 2011 |
Compositions and methods of use of borole derivatives, including benzoxaboroles, benzazaboroles and benzthiaboroles, as therapeutic agents for treatment of diseases caused by bacteria or viruses are disclosed, as well as methods for synthesis of said agents and compositions thereof.
Inventors: | Lee; Ving (Los Altos, CA), Plattner; Jacob J. (Berkeley, CA), Benkovic; Stephen J. (State College, PA), Baker; Stephen J. (Mountain View, CA), Maples; Kirk R. (San Jose, CA), Bellinger-Kawahara; Carolyn (Redwood City, CA), Akama; Tsutomu (Sunnyvale, CA), Zhang; Yong-Kang (San Jose, CA), Singh; Rajeshwar (Edmonton, CA), Sauro; Vittorio A. (Edmonton, CA) |
Assignee: |
Anacor Pharmaceuticals, Inc.
(Palo Alto,
CA)
|
Appl. No.: | 12/270,636 |
Filed: | November 13, 2008 |
Application Number | Filing Date | Patent Number | Issue Date | ||
10868268 | Jun., 2004 | 7465836 | |||
60478921 | Jun., 2003 | ||||
Current U.S. Class: | 568/8 |
Current International Class: | C07F 9/02 (20060101) |
5880188 | March 1999 | Austin et al. |
7465836 | December 2008 | Lee et al. |
2225014 | Jun., 1999 | CA | |||
WO 03033002 | Apr., 2003 | WO | |||
Genaev, A., et al., "Intramolecular Borylation Reaction Catalyzed by Lewis Acid: Preparation of 1H-2,1-Benzazaborole Derivatives", Chemical Communications, 2000, vol. 17; pp. 1587-1588. cited by other. |